Endralazine

Last updated
Endralazine
Endralazine.svg
Clinical data
ATC code
Identifiers
  • 6-benzoyl-3-hydrazinyl-5H,6H,7H,8H-pyrido[4,3-c]pyridazine
CAS Number
PubChem CID
ChemSpider
UNII
KEGG
ChEMBL
CompTox Dashboard (EPA)
Chemical and physical data
Formula C14H15N5O
Molar mass 269.308 g·mol−1
3D model (JSmol)
  • c1ccc(cc1)C(=O)N2CCc3c(c/c(=N/N)/[nH]n3)C2
  • InChI=1S/C14H15N5O/c15-16-13-8-11-9-19(7-6-12(11)17-18-13)14(20)10-4-2-1-3-5-10/h1-5,8H,6-7,9,15H2,(H,16,18) X mark.svgN
  • Key:ALAXZYHFVBSJKZ-UHFFFAOYSA-N X mark.svgN
 X mark.svgNYes check.svgY  (what is this?)    (verify)

Endralazine is an antihypertensive of the hydrazinophthalazine chemical class. [1] It is not approved for use in the United States.

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<span class="mw-page-title-main">Hydrazinophthalazine</span> Drug class

Hydrazinophthalazines are a class of antihypertensive drugs including:

References

  1. Meredith PA, Elliott HL, McSharry DR, Kelman AW, Reid JL (July 1983). "The pharmacokinetics of endralazine in essential hypertensives and in normotensive subjects". British Journal of Clinical Pharmacology. 16 (1): 27–32. doi:10.1111/j.1365-2125.1983.tb02139.x. PMC   1427948 . PMID   6882620.