Afurolol

Last updated
Afurolol
Afurolol.png
Clinical data
ATC code
  • none
Identifiers
  • 7-[3-(tert-Butylamino)-2-hydroxy-propoxy]-3H-isobenzofuran-1-one
CAS Number
PubChem CID
ChemSpider
UNII
ChEMBL
Chemical and physical data
Formula C15H21NO4
Molar mass 279.336 g·mol−1
3D model (JSmol)
  • O=C1OCc2cccc(OCC(O)CNC(C)(C)C)c12
  • InChI=1S/C15H21NO4/c1-15(2,3)16-7-11(17)9-19-12-6-4-5-10-8-20-14(18)13(10)12/h4-6,11,16-17H,7-9H2,1-3H3 Yes check.svgY
  • Key:NFXPPCYKSAAUMQ-UHFFFAOYSA-N Yes check.svgY
 X mark.svgNYes check.svgY  (what is this?)    (verify)

Alfurolol is a beta blocker. [1] [2]

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Monosaccharides, also called simple sugars, are the simplest form of sugar and the most basic units (monomers) of carbohydrates. The general formula is C
n
H
2n
O
n
, albeit not all molecules fitting this formula are carbohydrates. They are usually colorless, water-soluble, and crystalline solids. Contrary to their name (sugars), only some monosaccharides have a sweet taste.

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In chemistry, an enantiomer is one of two stereoisomers that are mirror images of each other that are non-superposable, much as one's left and right hands are mirror images of each other that cannot appear identical simply by reorientation. A single chiral atom or similar structural feature in a compound causes that compound to have two possible structures which are non-superposable, each a mirror image of the other. Each member of the pair is termed an enantiomorph ; the structural property is termed enantiomerism. The presence of multiple chiral features in a given compound increases the number of geometric forms possible, though there may still be some perfect-mirror-image pairs.

Zeppelin bend

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In geometry, a figure is chiral if it is not identical to its mirror image, or, more precisely, if it cannot be mapped to its mirror image by rotations and translations alone. An object that is not chiral is said to be achiral.

Chirality (chemistry) Geometric property of some molecules and ions

In chemistry, a molecule or ion is called chiral if it cannot be superposed on its mirror image by any combination of rotations and translations. This geometric property is called chirality. The terms are derived from Ancient Greek χείρ (cheir), meaning "hand"; which is the canonical example of an object with this property.

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Pheneturide

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Adaprolol is a beta blocker.

Ancarolol

Ancarolol is a beta blocker.

Arnolol

Arnolol is a beta blocker.

Xipranolol

Xipranolol is a beta blocker.

Xibenolol

Xibenolol is a beta blocker.

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Lorbamate

Lorbamate is a muscle relaxant and tranquilizer of the carbamate family which was never marketed.

Drug nomenclature is the systematic naming of drugs, especially pharmaceutical drugs. In the majority of circumstances, drugs have 3 types of names: chemical names, the most important of which is the IUPAC name; generic or nonproprietary names, the most important of which are the International Nonproprietary Names (INNs); and trade names, which are brand names. Under the INN system, generic names for drugs are constructed out of affixes and stems that classify the drugs into useful categories while keeping related names dinstinguishable. A marketed drug might also have a company code or compound code.

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References

  1. "The Use of Common Stems in the Selection of International Nonproprietary Names (INN) for Pharmaceutical Substances: Alphabetical list of stems together with corresponding INNs".
  2. Narimatsu S, Takemi C, Kuramoto S, Tsuzuki D, Hichiya H, Tamagake K, Yamamoto S (May 2003). "Stereoselectivity in the oxidation of bufuralol, a chiral substrate, by human cytochrome P450s". Chirality. 15 (4): 333–9. doi:10.1002/chir.10212. PMID   12666241.