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Names | |
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IUPAC name 4-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-4,5,6,7-tetrahydro-1,2-benzoxazol-3-one | |
Identifiers | |
3D model (JSmol) | |
ChEMBL | |
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Properties | |
C22H26N2O2S2 | |
Molar mass | 414.58 g·mol−1 |
Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa). |
EF-1502 is a GABA reuptake inhibitor. It could potentially be used to treat seizures.
EF-1502 has been shown to inhibit the type 1 GABA transporter (GAT1) [1] and the sodium and chloride-dependent betaine transporter (BGT-1). [2]
Tests in mice have shown that this compound possesses and anticonvulsant effect due to its GABA reuptake inhibiting properties. [3] [4]