Sulfametrole

Last updated
Sulfametrole
Sulfametrole.svg
Sulfametrole 3D spacefill.png
Clinical data
AHFS/Drugs.com International Drug Names
Routes of
administration
Oral
ATC code
Legal status
Legal status
  • In general: ℞ (Prescription only)
Identifiers
  • 4-amino-N-(4-methoxy-1,2,5-thiadiazol-3-yl)benzenesulfonamide
CAS Number
PubChem CID
ChemSpider
UNII
KEGG
ChEBI
ECHA InfoCard 100.046.611 OOjs UI icon edit-ltr-progressive.svg
Chemical and physical data
Formula C9H10N4O3S2
Molar mass 286.32 g·mol−1
3D model (JSmol)
  • COc1c(nsn1)NS(=O)(=O)c2ccc(cc2)N
  • InChI=1S/C9H10N4O3S2/c1-16-9-8(11-17-12-9)13-18(14,15)7-4-2-6(10)3-5-7/h2-5H,10H2,1H3,(H,11,13)
  • Key:IZOYMGQQVNAMHS-UHFFFAOYSA-N
   (verify)

Sulfametrole (INN) is a sulfonamide antibacterial.

It can be given with trimethoprim. [1]

Related Research Articles

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<span class="mw-page-title-main">Trimethoprim</span> Antibiotic

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Sulfadimidine or sulfamethazine is a sulfonamide antibacterial.

<span class="mw-page-title-main">Brodimoprim</span> Chemical compound

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Tetroxoprim (INN) is a derivative of trimethoprim. It was first described in 1979.

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Trimethoprim/sulfadoxine, sold under the brand name Trimidox, is an antibacterial agent that is used in cattle and swine to prevent and treat infections by both Gram-negative and Gram-positive bacteria.

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Isoniazid/pyridoxine/sulfamethoxazole/trimethoprim (INH/B6/CTX) is a fixed-dose combination medication for the prevention of opportunistic infections in HIV/AIDS. It combines isoniazid, pyridoxine, sulfamethoxazole, and trimethoprim. Specifically it is used to prevent tuberculosis, toxoplasmosis, pneumonia, malaria, and isosporiasis. It is taken by mouth.

Trimethoprim/sulfadiazine (TMP/SDZ) is a combination drug composed of trimethoprim and sulfadiazine used in the treatment of bacterial infections of animals, particularly horses.

References

  1. Plummer FA, Nsanze H, D'Costa LJ, et al. (July 1983). "Single-dose therapy of chancroid with trimethoprim-sulfametrole". N. Engl. J. Med. 309 (2): 67–71. doi:10.1056/NEJM198307143090202. PMID   6343878.