LY03017

Last updated
LY03017
Clinical data
Other namesLY-03017; LPM-526000133; LPM526000133
Routes of
administration
Oral [1] [2]
Drug class Serotonin 5-HT2 receptor antagonist; Serotonin 5-HT2A receptor inverse agonist; Serotonin 5-HT2C receptor antagonist

LY03017, also known as LPM-526000133, is a serotonin 5-HT2 receptor antagonist which is under development for the treatment of schizophrenia. [1] [3] [2] It acts specifically as a dual serotonin 5-HT2A receptor inverse agonist and serotonin 5-HT2C receptor antagonist. [1] [3] [2] The drug is under development by Luye Pharma Group in China. [1] [3] As of December 2025, it is in phase 1 clinical trials. [1] [3] [2] The chemical structure of LY03017 does not yet appear to have been disclosed. [1]

See also

References

  1. 1 2 3 4 5 6 "LY 03017". AdisInsight. 31 December 2025. Retrieved 31 January 2026.
  2. 1 2 3 4 "LY-03017 Drug Profile". Ozmosi. 1 January 1900. Retrieved 31 January 2026.
  3. 1 2 3 4 "Delving into the Latest Updates on LPM526000133 with Synapse". Synapse. 24 January 2026. Retrieved 31 January 2026.